Tolterodine Tartrate
Ponahalo | Tšoeu kapa hoo e ka bang tšoeu bonaleli phofo, odorless. |
Ho qhibiliha | Ho qhibiliha ka mokhoa o fokolang methapeng, e qhibilihang hanyane ka metsing, e sa qhibilihe ka har'a chloroform |
Qhibiliha | 205 ~ 2 10 ºC, e bole nakong ea ts'ebetso |
Potoloho e khethehileng | + 27.0º ~ + 30.0º |
Boitsebiso | |
Liketso tsa lik'hemik'hale | Tharollo e bonahala e ikemiselitse |
Ho monya litšobotsi | E bonts'a palo e kaholimo ho 282nm |
IR | Phallo ea IR ea tolterodin tartrate e lokela ho lumellana le seo (IR Album No. 1037) ea ntho e buuoang |
Seipone sa silevera se itšoara joang | Eketsa ammonia ea mokelikeli ka marotholi a silevera a nitrate a mangata, e kenye ka bateng ea metsi le mocheso, silevera ea arohana ebe e hokela leboteng le kahare la tube, seipone sa silevera |
Teko | |
Bohloko | PH: 3.0-4.5 |
Lhloride | Ha ea lokela ho ba matla ho feta resolution resolution e sebelisang 2.0ml ea sodium chloride standard solution (0.025%) |
Sulfate | Ha ea lokela ho ba matla ho feta resolutionolution e sebelisang 1.0ml ea potassium sulphate standard solution (0.05%) |
Laevo moqapi | NMT1.0% |
Lintho tse amanang | Ho se hloeke ho hong le ho hong: NMT0.1% |
Litšila tse felletseng: NMT 0.5% | |
Mosebetsi | Tolterodine ke mohanyetsi oa M ea amohelang tlholisano, 'me khetho ea eona ea senya e matla haholo ho feta tšoelesa ea salivary. Thibelo ea eona ea khutsufatso ea senya e makhetlo a ka bang 20 ho feta ea tšoelesa ea mathe. Kamora ho fana ka molomo oa tolterodine, sehlahisoa se ka sehloohong se sebetsang sa metabolite 5-hydroxymethyl (DD01) se hlahisoang ke sebete se ts'oana le ts'ebetso ea batsoali ea antimuscarinic mme se na le bohlokoa ba bohlokoa ba kalafo. Ka bobeli li na le kamano e nyane bakeng sa li-receptor tse ling tsa methapo ea kutlo le lipheo tse ka bang teng tsa lisele tse kang liteishene tsa calcium. |
Ngola molaetsa oa hau mona ebe u o romella ho rona