China Rifaximin ile-iṣẹ ati awọn olupese | Tecsun

Rifaximin

Apejuwe Kukuru:

Rifampicin (Rifaximin), a derivative of rifamycin, was developed by Alfa Italy. It was marketed in Italy as an anti-infectious diarrhea drug in 1987 and is still widely used abroad. Approved by SFDA in 2004, it has been used in clinical practice in China. It is a semi-synthetic antibacterial drug of rifamycin. It has a broad antibacterial spectrum and strong antibacterial activity. It can form a higher concentration of blood in the intestinal tract. It can inhibit Staphylococcus aureus, St...


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Rifampicin (Rifaximin), itọsẹ ti rifamycin, ni idagbasoke nipasẹ Alfa Italia. O ta ni Ilu Italia gẹgẹbi oogun igbẹ gbuuru alatako-arun ni 1987 ati pe o tun lo ni kariaye. Ti fọwọsi nipasẹ SFDA ni ọdun 2004, o ti lo ni iṣẹ iṣoogun ni Ilu China. O jẹ oogun antibacterial ologbele-sintetiki ti rifamycin. O ni iwoye antibacterial gbooro ati iṣẹ antibacterial lagbara. O le ṣe ifọkansi ifọkanbalẹ ti ẹjẹ ti o ga julọ ninu ara ifun. O le ṣe idiwọ Staphylococcus aureus, Streptococcus faecalis ati Salmonella ninu awọn eerobes ti o ni giramu-rere, eyiti o jẹ ti iru-ara Salmonella ni Giramu-odi aerobic kokoro arun. Shigella ati Escherichia coli, Yersinia enterocolitica ati Gram-positive anaerobic bacteria gbogbo wọn ni iṣẹ antibacterial giga. Ilana ti iṣe rẹ ni lati dojuti polymerase kokoro, dẹkun ilana transcription ti RNA, ati lẹhinna dẹkun kolaginni ti amuaradagba kokoro, nitorinaa dinku iṣelọpọ ti amonia. 1) iṣẹ antibacterial lagbara, ati iwoye antibacterial gbooro. O ni ipa ipakokoro lori ọpọlọpọ awọn giramu-rere awọn kokoro ati giramu ti ko ni giramu (pẹlu awọn kokoro aerobic ati awọn kokoro anaerobic), ati ipa lori awọn kokoro-giramu ti o dara giramu lagbara ju ti lọ lori kokoro-arun odi-giramu. 2) kii ṣe gba nipasẹ ọna ikun ati inu, ati pe ifọkansi rẹ ga gidigidi ninu iṣan inu. O le pa ajakalẹ-arun ti ara inu ati mu ipa egboogi-kokoro ni kiakia ni agbegbe agbegbe, ati pe ko ṣe pataki lati lo antispasmodic ati awọn oogun ipolowo ni apapo pẹlu apa ifun.

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