Carvedilol
Chigadzirwa zita | Carvedilol |
Chitarisiko | chena crystalline upfu, munhuwi |
Solubility | sungunuka mu glacial acetic acid; Soluble mu chloroform; Zvishoma zvinogadzikana mu methanol ethyl acetate; Inenge isinga nyungudike mumvura. |
Nzvimbo yakanyunguduka | 114.0 ~ 118.0ºC |
Chitupa | λmax = 285nm, 319nm, 331nm ± 2nm |
0.4-0.44 (iyo absorbance reshiyo ye331nm uye 285nm) | |
Infrared absorption spectrum inofanirwa kunge ichienderana nereferenzi chinhu | |
Kujeka uye ruvara rweacetic acid mhinduro | yakajeka uye isina ruvara, Max. Yero yero |
Singel kara mhinduro |
≤0.2% |
Yese tsvina | ≤0.5% |
Kurasikirwa pakuoma | ≤0.5% |
Residue pamusoro kuvesa | ≤0.1% |
basa | Carvedilol ine moyo wakasimba uye neuroprotective mhedzisiro: kusiyana neyakajairwa β-receptor vanopikisa, kushandiswa kwenguva refu kwechigadzirwa ichi mune varwere vane hutachiona hwakanyanya hakugone chete kudzora coronary uye renal midziyo, kudzora peripheral vascular kuramba, asi zvakare kuderedza systemic kutenderera. Uye pulmonary kutenderera kuramba, zvinobudirira kudzora yakakwira BP. Ichi chigadzirwa chine chekudzivirira pabasa renal, hachinje renal kuyerera kweropa, asi chinoderedza microalbuminuria, inoderedza renal vascular kuramba, uye ine yakanaka yekumisikidza mhedzisiro paropa lipids. |
Nyora yako meseji pano uye uitumire kwatiri