Carvedilol
Ingoa hua | Carvedilol |
Te Ahua | paura tioata ma, kore haunga |
Te wairewa | wairewa i roto i te waikawa ahetiki hukapapa; He wairewa i te chloroform; He iti nei te wairewa i te methanol ethyl acetate; Kaore e rewa i te wai. |
Wāhi rewa | 114.0 ~ 118.0ºC |
Tuakiri | λmax = 285nm, 319nm, 331nm ± 2nm |
0.4-0.44 (te ōwehenga mimiti o 331nm me 285nm) | |
Kia rite ki te matū tohutoro te hihinga hihinga ngongo pungarehu | |
Maama me te tae o te waikawa waikawa acetic | maama me te kore tae, Max. Kōwhai paerewa |
Te color solution |
≤0.2% |
Tapeke poke | ≤0.5% |
Ngaronga o te maroke | ≤0.5% |
Toenga i runga i te mura | ≤0.1% |
mahi | He kaha te ngakau o te Carvedilol me nga awangawanga neuroprotective: kaore i rite ki nga kaitautoko β-kaiwhiwhi noa, ko te whakamahinga mo te wa roa o tenei hua ki nga tuuroro haumanu kaore e taea te whakarake i nga kawa o te kawa me nga whatukuhu, ka whakaheke i te aukati auroro, engari ka whakaiti ano hoki i te tohanga o te punaha. Me te aukati tohanga porohita, ka tino whakahaere i te toto toto tiketike. Ko tenei hua he aarai ki runga i te mahi whatukuhu, kaore e rereke te rere o te toto, engari ka whakaheke i te microalbuminuria, ka whakaitihia te awangawanga o te whatukuhu, ka pai te whakahaere ki nga lipid toto. |
Tuhia to korero ki konei ka tuku mai ki a maatau