Carvedilol
Aha ngwaahịa | Carvedilol |
Ọdịdị | ọcha crystalline ntụ ntụ, odorless |
Solubility | soluble na glacial acetic acid; Soluble na chloroform; Ntucha soluble na methanol ethyl acetate; Ihe anaghị edozi na mmiri. |
Ebe mgbaze | 114.0 ~ 118.0ºC |
Njirimara | max = 285nm, 319nm, 331nm ± 2nm |
0.4-0.44 (njedebe nke 331nm na 285nm) | |
Infrared absorption dị iche iche kwesịrị ikwekọ na ntinye ihe | |
Ihe doro anya na agba nke ngwọta acetic acid | doro anya na enweghị ntụpọ, Max. Ọkọlọtọ edo edo |
Singel color solution |
≤0.2% |
Total adịghị | 0.5% |
Loss na ihicha | 0.5% |
Fọduru na mgbanye | ≤0.1% |
ọrụ | Carvedilol nwere obi siri ike na mmetụta neuroprotective: n'adịghị ka ndị na-emegide β-receptor nkịtị, iji ngwaahịa a ogologo oge na ndị ọrịa na-arịa ọbara mgbali elu nwere ike ọ bụghị naanị ịbawanye akwara na akwara akwara, belata nguzogide vascular elu, kamakwa belata usoro mgbasa. Na akpa ume mgbasa eguzogide, n'ụzọ dị irè ịchịkwa ọbara mgbali elu. Ngwaahịa a nwere mmetụta nchedo na arụmọrụ nke akụrụ, anaghị agbanwe nsụgharị akụrụ, ma na-ebelata microalbuminuria, na-ebelata nguzogide akwara akụrụ, ma nwee usoro nchịkwa dị mma na lipids ọbara. |
Dee ozi gị ebe a ma zitere anyị ya