Carvedilol
Khoom npe | Carvedilol |
Tsos | dawb crystalline hmoov, ntxhiab tsw |
Tub sab | soluble hauv glacial acetic acid; Soluble hauv chloroform; Me ntsis soluble hauv methanol ethyl acetate; Siv cov tshuaj tsis haum rau dej. |
Melting taw tes | 114.0 ~ 118.0ºC |
Tus Kheej | max = 285nm, 319nm, 331nm ± 2nm |
0.4-0.44 (qhov nqus piv ntawm 331nm thiab 285nm) | |
Infrared absorption spectrum yuav tsum muaj raws li cov khoom siv tshuaj | |
Clarity thiab xim ntawm cov kua tshuaj acetic acid | ntshiab thiab tsis muaj xim, Max. Txuj daj |
Singel xim daws |
≤0.2% |
Tag nrho impurities | 0.5% |
Poob rau kom qhuav | 0.5% |
Residue ntawm kev tiv thaiv | ≤0.1% |
muaj nuj nqi | Carvedilol muaj lub plawv muaj zog thiab mob neuroprotective: tsis zoo li ib txwm β-receptor antagonists, kev siv lub sijhawm ntev ntawm cov khoom no hauv cov neeg mob ntshav siab tsis tuaj yeem tsis tsuas yog txhim kho cov hlab plawv thiab cov hlab ntsha hauv lub plawv, txo cov leeg kev tawm tsam, tab sis kuj txo cov kev tiv thaiv kab ke. Thiab pulmonary ncig tsis kam, zoo tswj ntshav siab. Cov khoom no muaj kev tiv thaiv rau lub raum kev ua haujlwm, tsis hloov ntshav hloov pauv, tab sis txo microalbuminuria, txo cov roj ntsha raum tsis kam, thiab muaj cov kev cai tswj tau zoo ntawm cov ntshav lipids. |
Sau koj cov lus ntawm no thiab xa rau peb