ʻO Carvedilol
Inoa mea kūʻai | ʻO Carvedilol |
Helehelena | pauka aniani keʻokeʻo, ʻaʻohe onaona |
Solubility | wailana i ka glacial acetic acid; Wehe i loko o ka chloroform; Hiki ke hoʻoheheʻe iki ʻia i ka methanol ethyl acetate; Hoʻomaʻemaʻe ʻole ʻia i ka wai. |
Kuhi hoʻoheheʻe | 114.0 ~ 118.0ºC |
ʻIʻike | λmax = 285nm, 319nm, 331nm ± 2nm |
0.4-0.44 (ka lakio absorbance o 331nm a me 285nm) | |
Pono e kūlike me ka mea kuhikuhi | |
Ke akāka a me ke kala o ka hopena acid acetic | mōakāka a kala ʻole, Max. Melemele maʻamau |
ʻO color solution |
≤0.2% |
Huina haumia | ≤0.5% |
Lilo i ka hoʻomaloʻo ʻana | ≤0.5% |
Koena ma ka hoʻā ʻana | ≤0.1% |
hana | Loaʻa ka puʻuwai ikaika a me nā hopena neuroprotective ʻo Carvedilol: ʻokoʻa ka antagonists β-receptor maʻamau, hoʻohana lōʻihi o kēia huahana i nā mea maʻi hypertensive ʻaʻole hiki ke hoʻonui i nā moku coronary a me nā puʻuwai, hōʻemi i ke kūpaʻa vipher peripheral, akā hoʻoliʻiliʻi hoʻi i ka ʻōnaehana ʻōnaehana. A me ke kūpaʻa o ka pulmonary, e kāohi pono i ke kaomi kiʻekiʻe. He hopena pale kā kēia huahana ma ka hana renal, ʻaʻole ia e loli i ke kahe o ke kōkō, akā hoʻemi ʻia ka microalbuminuria, hoʻoliʻiliʻi i ke kūpaʻa venal a me ka hopena maikaʻi o ke kaohi i nā lipids koko. |
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