Carvedilol
Igoa oloa | Carvedilol |
Foliga Vaaia | efuefu crystalline paʻepaʻe, leai se manogi |
Solubility | soluble i glacial acetic acid; Soluble i le chloroform; Laʻititi soluble i methanol ethyl acetate; E masani ona le mafai ona sosolo i le vai. |
Faaliusuavai | 114.0 ~ 118.0ºC |
Faʻailoaina | λmax = 285nm, 319nm, 331nm ± 2nm |
0.4-0.44 (o le fua faʻatusatusa o le 331nm ma le 285nm) | |
E tatau ona ogatasi le fusi o alaleo faʻaafa ma fua o faʻamatalaga | |
Malamalama ma lanu o le acetic acid solution | manino ma leai se lanu, Max. Lanu samasama |
Singel color solution |
≤0.2% |
Aofai o mea le mama | ≤0.5% |
Maliu i le mago | ≤0.5% |
Toe totoe i luga o le afi | ≤0.1% |
gaioiga | O le Carvedilol e malosi lona fatu ma aʻafiaga o le neuroprotective: e le pei o le masani β-receptor antagonists, o le faʻaaoga umi o lenei oloa i tagata mamaʻi e le gata e mafai ai ona faʻalauteleina vaʻaia ma fatugaʻo vaʻa, faʻaititia vafeagai teteega, ae faʻaititia foʻi le faʻataʻamilosaga. Ma tetee teteʻe pulmonary, lelei pulea maualuga toto maualuga. Lenei oloa ei ai se aafiaga puipuia i gaioiga fatugao, e le suia renal toto tafe, ae faaititia microalbuminuria, faaitiitia Fatugao tetee tetee, ma ei ai se lelei tulafono faatonutonu aafiaga i le toto lipids. |
Tusi lau feʻau ii ma lafo mai ia matou