China Carvedilol ifektri abakhiqizi | UTecsun

ICarvedilol

Incazelo emfushane:

Product name Carvedilol Appearance white crystalline powder,odourless Solubility soluble in glacial acetic acid;Soluble in chloroform;Slightly soluble in methanol ethyl acetate;Practically insoluble in water. Melting point 114.0~118.0ºC Identification λmax=285nm,319nm,331nm±2nm 0.4-0.44(the absorbance ratio of 331nm and 285nm) Infrared absorption spectrum should be consistent with the reference substance Clarity and color of acetic acid solution clear and colorless ,...


Imininingwane yomkhiqizo

Amathegi womkhiqizo

Igama lomkhiqizo ICarvedilol
Ukubukeka impuphu emhlophe emhlophe, engenaphunga
Ukuncibilika encibilikayo e-glacial acetic acid; Encibilikayo ku-chloroform; Encibilikayo kancane ku-methanol ethyl acetate; Cishe ayincibiliki emanzini.
Iphuzu lokuncibilika 114.0 ~ 118.0ºC
Umazisi λmax = 285nm, 319nm, 331nm ± 2nm
0.4-0.44 (isilinganiso sokumunca esingu-331nm nesingu-285nm)
I-infrared absorption spectrum kufanele ihambisane nento yokubhekisela
Ukucaca nombala  acetic acid icacile futhi ayinambala, uMax. Okuphuzi okujwayelekile
Singel
color solution
≤0.2%
Ukungcola okuphelele ≤0.5%
Ukulahlekelwa kokomiswa ≤0.5%
Izinsalela zokushisa ≤0.1%
umsebenzi I-Carvedilol inemiphumela eqinile yenhliziyo kanye ne-neuroprotective: ngokungafani nabaphikisi abajwayelekile be-β-receptor, ukusetshenziswa kwesikhathi eside kwalo mkhiqizo ezigulini ezinomfutho wegazi ophezulu akukwazi nje kuphela ukukhulisa imikhumbi ye-coronary ne-renal, kunciphise ukumelana nemithambo yegazi, kepha futhi kunciphise ukusakazwa kwesistimu. Futhi ukumelana nokujikeleza kwamaphaphu, kulawula ngempumelelo umfutho wegazi ophezulu. Lo mkhiqizo unomphumela wokuvikela ekusebenzeni kwezinso, awuguquki ukugeleza kwegazi le-renal, kepha wehlisa i-microalbuminuria, wehlise ukumelana nemithambo yegazi, futhi unomphumela omuhle wokulawula kuma-lipids egazi.

 

 


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