ICarvedilol
Igama lomkhiqizo | ICarvedilol |
Ukubukeka | impuphu emhlophe emhlophe, engenaphunga |
Ukuncibilika | encibilikayo e-glacial acetic acid; Encibilikayo ku-chloroform; Encibilikayo kancane ku-methanol ethyl acetate; Cishe ayincibiliki emanzini. |
Iphuzu lokuncibilika | 114.0 ~ 118.0ºC |
Umazisi | λmax = 285nm, 319nm, 331nm ± 2nm |
0.4-0.44 (isilinganiso sokumunca esingu-331nm nesingu-285nm) | |
I-infrared absorption spectrum kufanele ihambisane nento yokubhekisela | |
Ukucaca nombala acetic acid | icacile futhi ayinambala, uMax. Okuphuzi okujwayelekile |
Singel color solution |
≤0.2% |
Ukungcola okuphelele | ≤0.5% |
Ukulahlekelwa kokomiswa | ≤0.5% |
Izinsalela zokushisa | ≤0.1% |
umsebenzi | I-Carvedilol inemiphumela eqinile yenhliziyo kanye ne-neuroprotective: ngokungafani nabaphikisi abajwayelekile be-β-receptor, ukusetshenziswa kwesikhathi eside kwalo mkhiqizo ezigulini ezinomfutho wegazi ophezulu akukwazi nje kuphela ukukhulisa imikhumbi ye-coronary ne-renal, kunciphise ukumelana nemithambo yegazi, kepha futhi kunciphise ukusakazwa kwesistimu. Futhi ukumelana nokujikeleza kwamaphaphu, kulawula ngempumelelo umfutho wegazi ophezulu. Lo mkhiqizo unomphumela wokuvikela ekusebenzeni kwezinso, awuguquki ukugeleza kwegazi le-renal, kepha wehlisa i-microalbuminuria, wehlise ukumelana nemithambo yegazi, futhi unomphumela omuhle wokulawula kuma-lipids egazi. |
Bhala umyalezo wakho lapha bese uwuthumela kithi