Ulbenimex
Inoa huahana : | ʻO Ubenimex |
MF: | C 16H 24N 2O 4 |
CAS NO: | 73334-07-3 |
Helehelena: | ʻO ka pauka crystalline keʻokeʻo, ʻaʻohe onaona, ʻono ʻawaʻawa, ʻoluʻolu hikiwawe ʻia i ka waikawa acetic, hiki ke hoʻoheheʻe ʻia i ka wai a me ka methanol, hiki ke hoʻoheheʻe ʻia i ka waikawa hydrochloric a me Sodium hydroxide |
ʻAno Molecular |
1, hele mai ia mai Streptomyces olivoreticuli
2, He hoʻokūkū kēia, a me nā mea hoʻohuli protease hiki ke hoʻohuli ʻia.
3, Loaʻa iā ia kahi hopena inhibitory ma arginylaminopeptidase, leukotriene A4 hydrolase, alanyl aminopeptidase, a me leucyl / cyanoamido peptidase.
4, hiki i kēia huahana ke hoʻonui i ka hana pale, i hoʻohana ʻia no ka chemotherapy anti-cancer, hana hoʻomaʻamaʻa adjuvant o radiotherapy, nā kīnā ʻole immune senile. Hiki ke hoʻohui ʻia me chemotherapy, radiotherapy a me ka hoʻopili ʻana i ka leukemia, myeloma maha, myelodysplastic syndrome a me ka transplantation cell hematopoietic, a me nā mea maʻi tumo paʻa ʻē aʻe.
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